Ex Parte Kneen et alDownload PDFPatent Trial and Appeal BoardFeb 16, 201611629982 (P.T.A.B. Feb. 16, 2016) Copy Citation UNITED STA TES p A TENT AND TRADEMARK OFFICE APPLICATION NO. FILING DATE FIRST NAMED INVENTOR 111629,982 11/01/2007 26111 7590 02/17/2016 STERNE, KESSLER, GOLDSTEIN & FOX P.L.L.C. 1100 NEW YORK A VENUE, N.W. WASHINGTON, DC 20005 GeoffKneen UNITED STATES DEPARTMENT OF COMMERCE United States Patent and Trademark Office Address: COMMISSIONER FOR PATENTS P.O. Box 1450 Alexandria, Virginia 22313-1450 www .uspto.gov ATTORNEY DOCKET NO. CONFIRMATION NO. 2400.1340000/RWE/SLE 1111 EXAMINER BROWN, COURTNEY A ART UNIT PAPER NUMBER 1617 MAILDATE DELIVERY MODE 02/17/2016 PAPER Please find below and/or attached an Office communication concerning this application or proceeding. The time period for reply, if any, is set in the attached communication. PTOL-90A (Rev. 04/07) UNITED STATES PATENT AND TRADEMARK OFFICE BEFORE THE PATENT TRIAL AND APPEAL BOARD Ex parte GEOFF KNEEN, ANNE SUTY-HEINZE, PETER DAHMEN, YASUO ARAKI, TAKUMA SHIGYO, and HANS-LUDWIG ELBE Appeal2013-004485 Application 11/629,982 Technology Center 1600 Before DEMETRA J. MILLS, JOHN G. NEW, and ROBERT A. POLLOCK, Administrative Patent Judges. MILLS, Administrative Patent Judge. DECISION ON APPEAL This is an appeal under 35 U.S.C. § 134. The Examiner has rejected the claims for obviousness. We have jurisdiction under 35 U.S.C. § 6(b). We affirm. Appeal2013-004485 Application 11/629,982 STATEMENT OF CASE According to the Specification, the "active compounds according to the invention have very good fungicidal properties and, in seed treatment, are particularly suitable for controlling phytopathogenic fungi, such as Ascomycetes and Basidiomycetes." Spec. 14. The following claim is representative. 7. A method of dressing seed for controlling Rhizoctonia solani comprising: treating said seed with N-[2-(l ,3-dimethylbutyl)phenyl]-5- fluoro-1,3-dimethyl- lH-pyrazole-4-carboxamide (I-2) at a rate of from 1 g to 50 g per 100 kg of seed, wherein said seed is rice seed. Cited References Elbe et al. Elbe et al. US 2004/0204470 Al Oct. 14, 2004 (hereinafter "Elbe '4 70") WO 03/010149 Al Feb. 6, 2003 (hereinafter "Elbe '149") Howell et al., Induction of Terpenoid Synthesis in Cotton Roots and Control of Rhizoctonia solani by Seed Treatment with Trichoderma virens, 90 PHYTOPATHOLOGY 248-252 (2000) (hereinafter "Howell"). Application No. 11/912,773 (hereinafter '773) Application No. 12/831,990 (hereinafter '990) Grounds of Rejection 1. Claims 7, 8, 15, 29, 33 and 34 are rejected under 35 U.S.C. § 103(a) as being unpatentable over Elbe' 149 (see equivalent translated document (Elbe '470)) in view of Howell. 2 Appeal2013-004485 Application 11/629,982 2. Claim 7 is provisionally rejected on the ground of nonstatutory obviousness-type double patenting as being unpatentable over claims 4 and 13 of copending Application No. 11/912,773. 3. Claim 7 is provisionally rejected on the ground of nonstatutory obviousness-type double patenting as being unpatentable over claim 1 of copending Application No. 12/831,990. FINDINGS OF FACT The Examiner's findings of fact (FF) are set forth in the Final Action dated April 25, 2012, pages 3-15 and Answer at pages 2-12. The following facts are highlighted. 1. Elbe '4 7 0 teaches the compound of instant formula I-a wherein R=hydrogen, R 1=hydrogen, R2=methyl, R3=methyl and R4=fluorine (see compound 1-21 (N-[2-(l,3-dimethylbutyl)phenyl]-5-fluoro-1,3- dimethyl- lll-pyrazole-4-carboxamide) [penflufen] on page 20, [0041] of corresponding document, US 2004/0204470). Ans. 9. 2. Elbe '470 teaches that the active compounds can be used in compositions to treat all plants and parts of plants which are to be understood as meaning all above-ground and below-ground parts and organs of plants, such as fruits and seeds and also roots, tubers and rhizomes as well as harvested plants and vegetative and generative propagation material, for example seedlings, tubers, rhizomes, cuttings and seeds (see i-f 224). Ans. 9. 3. Elbe '470 teaches (i-f 385) that the transgenic plants or plant cultivars which are preferably treated according to their invention include important crop plants, such as cereals (wheat, rice), maize, soya 3 Appeal2013-004485 Application 11/629,982 beans, potatoes, cotton (i-f 3 85). Ans. 9. 4. In addition, Elbe [ '4 7 0] teach[ es] that the compounds of the formula (I) according to their invention also have very good antimycotic activity. They have a very broad antimycotic activity spectrum in particular against dermatophytes and yeasts, molds and diphasic fungi, (for example against Candida species, such as Candida albicans, Candida glabrata ), and Epidermophyton jloccosum, Aspergillus species, such as Aspergillus niger and Aspergillus fumigatus, Trichophyton species, such as Trichophyton mentagrophytes, Microsporon species such as Microsporon canis and audouinii. The list of these fungi by no means limits the mycotic spectrum covered, but is only for illustration. i1379; Final Act. 10. 5. "Elbe ['470] teach[ es] that the list of these fungi by no means limits the mycotic spectrum covered, but is only for illustration ([0379]). For seed dressing, the active compound application rates are generally between 0.001 and 50 g per kilogram of seed, preferably between 0.01 and 10 g per kilogram of seed ([0381 ])." Final Act. 10. 6. "Depending on the plant species or plant cultivars, Elbe et al. teach[ es] their location and growth conditions (soils, climate, vegetation period, and diet), the treatment according to their invention may also result in super additive ('synergistic') effects ([0384]." Final Act. 10. 7. Elbe '4 70 discloses that the substances according to the invention "have potent microbicidal activity and can be employed for controlling undesirable microorganisms, such as fungi and bacteria, in 4 Appeal2013-004485 Application 11/629,982 crop protection and in the protection of material." i-f 184. "Fungicides can be employed in crop protection for controlling Plasmodio- phoromycetes, Oomycetes, Chytridiomycetes, Zygomycetes, Ascomycetes, Basidiomycetes1 and Deuteromycetes." i-f 185 (emphasis added). 8. Howell teaches that the Rhizoctonia solani is a well-known fungus which infects cotton seed. Abstract. 9. Howell discloses that it is well known to treat or dress cotton seed to control Rhizoctonia solani fungal infection. Abstract; Final Action 10. 10. Howell treats cotton seed with Trichoderma virens to control Rhizoctonia solani fungal infection of cotton seed. Abstract. PRINCIPLES OF LAW In making our determination, \'l.;e apply the preponderance of the evidence standard. See, e.g., Ethicon, Inc. v. Quigg, 849 F.2d 1422, 1427 (Fed. Cir. 1988) (explaining the general evidentiary standard for proceedings before the Office). The Board "determines the scope of claims in patent applications not solely on the basis of the claim language, but upon giving claims their broadest reasonable construction 'in light of the specification as it would be interpreted by one of ordinary skill in the art.'" Phillips v. AWH Corp., 415 F.3d 1303, 1316 (Fed. Cir. 2005) (quoting Jn re Am. Acad. of Sci. Tech. Ctr., 367 F.3d 1359, 1364 (Fed. Cir. 2004). 1 Rhizoctonia solani is a basidiomycete. http://www.extento.hawaii.edu/kbase/crop/type/r_solani.htm 5 Appeal2013-004485 Application 11/629,982 "In rejecting claims under 35 U.S.C. § 103, the examiner bears the initial burden of presenting a prima facie case of obviousness. Only if that burden is met, does the burden of coming forward with evidence or argument shift to the applicant." In re Rijckaert, 9 F.3d 1531, 1532 (Fed. Cir. 1993) (citations omitted). In order to determine whether a prima facie case of obviousness has been established, we consider the factors set forth in Graham v. John Deere Co., 383 U.S. 1, 17 (1966): (1) the scope and content of the prior art; (2) the differences between the prior art and the claims at issue; (3) the level of ordinary skill in the relevant art; and ( 4) objective evidence of nonobviousness, if present. "The combination of familiar elements according to known methods is likely to be obvious when it does no more than yield predictable results." KSR Int'! Co. v. Teleflex Inc., 550 U.S. 398, 416 (2007). In KSR, the Supreme Court also addressed the "obvious to try" issue: \X/hen there is a design need or market pressure to solve a problem and there are a finite number of identified, predictable solutions, a person of ordinary skill has good reason to pursue the known options within his or her technical grasp. If this leads to the anticipated success, it is likely the product not of innovation but of ordinary skill and common sense. In that instance the fact that a combination was obvious to try might show that it was obvious under § 103. Id. at 421. A prior art patent disclosed genus of 1200 effective combinations of compounds, including the claimed combination. It was held that the "[ d]isclos[ ure of] a multitude of effective combinations does not render any 6 Appeal2013-004485 Application 11/629,982 particular formulation less obvious." Merck & Co., v. Biocraft Labs. Inc., 874 F.2d 804, 807 (Fed. Cir. 1989). Rejection 1- Obviousness We agree with the Examiner's fact finding, statement of the rejection and responses to Appellants' arguments as set forth in the Final Action and Answer. We find that the Examiner has provided evidence to support a prima facie case of obviousness. We provide the following additional comment to the Examiner's argument set forth in the Final Action and Answer. With respect to the Examiner's prima facie case of obviousness, Appellants contend that: in view of Elbe, one would have to try all of the 54 individual pyrazolylcarboxanilides with all "compounds used to control fungi" disclosed in the art against all parts of plants disclosed in the art. This is not the "finite number of identified solutions" that would have made the invention obvious to try, and therefore obvious under 35 U.S.C. § 103. App. Br. 22-23. We are not persuaded. Elbe '470 specifically teaches the claimed antifungal compound, penflufen, compound I-21, page 20. Elbe '4 70 teaches that penflufen is a known fungicide which can be used for the treatment of fungal infections which include basidiomycete fungal infections. FF7. Elbe '4 70 teaches that their disclosed pyrazolylcarbox- anilides can be used to treat fungal infections of cotton and rice, and that seeds may be treated with their antifungal compounds, including penflufen. FF3, 5. While not specifically disclosing the fungal strain Rhizoctonia solani, Elbe '470 discloses that the provided list of fungi which can be 7 Appeal2013-004485 Application 11/629,982 treated with their pyrazolylcarboxanilides compounds "by no means limits the mycotic spectrum covered, but is only for illustration." Elbe '470 i-f379. Howell discloses that Rhizoctonia solani is known to infect cotton and that it is known in the art to treat cotton seed with antifungals against Rhizoctonia Solani. Therefore, we conclude that it would have been obvious to one of ordinary skill in the art at the time of the invention to use penflufen as an antifungal to address fungal infections of rice and cotton plants and to dress the seed of the rice and cotton plants with the antifungal, penflufen. The disclosure a multitude of effective fungal compounds in Elbe '4 7 0 does not render any particular fungal compound less obvious. Merck & Co., 87 4 F .2d at 807. Moreover, when there is a market pressure to solve a problem such as fungal infection of crop plants and there are a finite number of identified, predictable solutions, such as the use of a known penflufen fungicide, a person of ordinary skill has good reason to pursue the known options within his or her technical grasp. If this leads to the anticipated success, it is likely the product not of innovation but of ordinary skill and common sense. In that instance the fact that a combination was obvious to try might show that it was obvious under§ 103. KSR, 550 U.S. at 421. Appellants have presented no evidence that one of ordinary skill in the art would not have expected broad spectrum fugicidal activity from the penflufen fungicide disclosed in Elbe '470, including fungicidal activity against basidiomycete infections disclosed therein. FF7. Appellants also argue that they have provided clear evidence of unexpected results to rebut any prima facie case of obviousness presented by the Examiner. App. Br. 23. In particular, Appellants rely on data of 8 Appeal2013-004485 Application 11/629,982 unexpected results presented in the Declaration of Dr. Daniela Portz dated May 17, 2011. Dr. Portz Declaration provides the following Table at page 3. The Table compares efficacy of penflufen (compound disclosed in Elbe '470 and presently claimed) for the treatment of Rhizoctonia solani infection of cotton seed as compared with another antifungal compound of similar structure. Notably, the Table 3 example does not show the treatment of Rhizoctonia solani infection of rice seed, as claimed, and penflufen (bottom compound in Table) is clearly disclosed in Elbe '470. Therefore it is not immediately clear how the Portz Declaration provides unexpected results for the treatment of rice infection by Rhizoctonia solani. Moreover, even if Appellants had provided a clear explanation of the relevance of the Portz Table data to Rhizoctonia solani infection of rice seed, we agree with the Examiner that Appellants have not adequately explained how the data in the Portz Declaration is commensurate in scope with the rate of seed application claimed. Ans. 15. For example, Table C from the 9 Appeal2013-004485 Application 11/629,982 Specification, page 31, the only table of record which addresses data with respect to Rhizoctonia solani infection of rice, shows efficacy of the application of 200g/1 OOkg of seed, which is outside the claimed range of 1 to 50 g/lOOkg of rice seed. With respect to claim 15 and its dependent claims, notwithstanding any improper previous indication by the Examiner that there may have been a showing of unexpected results for a range of seed application within the claims (App. Br. 10), a preponderance of the evidence does not support Appellants' position and the obviousness rejection of the rejected claims is affirmed for the reasons of record and herein. Rejection 2-0bviousness-type Double Patenting '773 Claim 7 is provisionally rejected on the ground of nonstatutory obviousness-type double patenting as being unpatentable over claims 4 and 13 of copending Application No. 11/912,773. Claims 4 and 13 of copending Application No. 11/912,7732 are reproduced below. 4. A composition comprising a synergistic active compound 10 Appeal2013-004485 Application 11/629,982 combination, which comprises N-[2-( 1,3-dimethylbutyl)phenyl]-5-fluoro- 1,3-dimethyl- lH-pyrazole- 4-carboxamide having the following formula: H3C O N~-~ I N H I '--\// N H3C F H3C CH3 and one or more active compounds selected from the group consisting of (2 .1.1) clothianidin, (2.1.2) imidacloprid, (2.1.3) thiacloprid, (2 .1.4) thiamethoxam, (2. 1. 5) acetamiprid, (2 .1. 6) dinotefuran, (2 .1. 7) nitenpyram, nithiazine, (3 .1.1) methiocarb, (3 .1.2) thiodicarb, benfuracarb, carbosulfan, ( 4.1.1) beta-cyfluthrin, bifenthrin, cypermethrin, tefluthrin, transfluthrin. (5.1.1) spinosad, ( 6.2.1) fipronil, (6.2.2) ethiprole, avermectin, and (21.1.1) N2-[l, 1-dimethyl-2-(methylsulphonyl)ethyl]-3-iodo-N1-[2-methyl- 4-[ 1,2,2,2-tetrafluoro-l-( trifluoromethyl)ethyl]phenyl]-1,2-benzene- dicarboxamide, wherein the weight ratio ofN-[2-(l,3-dimethylbutyl)phenyl]- 5-fluoro-1,3-dimethyl-lH-pyrazole-4-carboxamide to said one or more active compounds is from 500:1to1:1000. 11 Appeal2013-004485 Application 11/629,982 13. A method of treating seeds, comprising contacting said seeds with the composition according to Claim 4. The Examiner argues that Copending Application No. 11/912,773 (hereinafter '773) and the instant application recite the same method of treating seeds using the compound formula I-a. However, the difference between the invention of the instant application and that of copending '773 is that the instant application does not require the use of a second active compound. However, it is known in the art that combining pesticides increase the efficacy of a pesticide such that the maximum level of control or pest control for a given application rate of a pesticide is increased, or alternatively, the application rate of a pesticide giving optimum control or pest control can be reduced. The Examiner maintains that one would have been motivated not to use a second active compound when an increase the efficacy of I-a is not desired. From this extensive overlap of subject matter, one of ordinary skill in the art would recognize that the same method is taught in copending application '773. Ans. 2-3. The Appellants argue that the Examiner impermissibly considered the disclosure of the '773 application. We are not persuaded. The record adequately reflects that Examiner here has compared the claims of the pending application to those of the '773 application. The Examiner is arguing that both sets of claims recite the same method of treating seeds in similar amounts using the compound formula I-a, penflufen. Be that as it may, we do find the Examiner's obviousness-type double patenting rationale deficient, in that the Examiner fails to provide evidence on this record to support the argument that 12 Appeal2013-004485 Application 11/629,982 it is known in the art that combining pesticides increase the efficacy of a pesticide such that the maximum level of control or pest control for a given application rate of a pesticide is increased, or alternatively, the application rate of a pesticide giving optimum control or pest control can be reduced. The Examiner maintains that one would have been motivated not to use a second active compound when an increase the efficacy of I-a is not desired. Ans. 2-3. While the Examiner could have cited a reference to support these arguments, she did not. We are constrained to reverse this rejection. The obviousness-type double patenting rejection over '773 is reversed. Rejection 3 - Obviousness-type Double Patenting '990 Claim 7 of the present application is provisionally rejected on the ground of nonstatutory obviousness-type double patenting as being unpatentable over claim 1 of copending Application No. 12/831,990. Claim 1 of the '990 application as amended July 14, 2015, is reproduced below. 1. A method for promoting early emergence of a crop, comprising applying to one or more seeds in need thereof a compound of formula (I) (I) in an amount effective to promote the early emergence 13 Appeal2013-004485 Application 11/629,982 of crops, wherein the crop is a soybean crop or a potato crop and wherein the seed is treated in absence of a pest pressure. The Examiner argues that: The copending application and the instant application recite the same method of treating seeds using the compound of I-a of the instant application. The difference between the invention of the instant application and that of copending '990 is that the instant application is drawn to a method for dressing seed and copending '990 is drawn to a method for increasing seedling growth and early emergence of a crop. However, both methods comprise dressing seed. From this extensive overlap of subject matter, one of ordinary skill in the art would recognize that the same method is taught in copending application '990. Final Act. 4--5. Appellants contend, "that it does not necessarily follow that practicing a method of claim 1 of the '990 application will control Rhizoctonia solani because the fungus may not be present." Reply Br. 7. \Ve are not persuaded by 1A .. ppellants' argument. "It is a general rule that merely discovering and claiming a new benefit of an old process cannot render the process again patentable." In re Woodruff, 919 F. 2d 1575, 1578 (Fed. Cir. 1990). It is also well settled that discovery of a property inherent to a prior art process does not render that process patentable, even if the prior art did not appreciate the property. Verdegaal Bros. Inc. v. Union Oil Co., 814 F.2d 628, 633 (Fed. Cir. 1987). However, "a limitation or the entire invention is inherent and in the public domain if it is the 'natural result flowing from' the explicit disclosure of the prior art." Schering Corp. v. Geneva Pharms., Inc., 339 F.3d 1373, 1379 (Fed. Cir. 2003). Pending claims either "read on" or do not "read on" the prior art. Kalman v. Kimberly-Clark Corp., 713 F.2d 760, 772 (Fed. Cir. 1983). In the 14 Appeal2013-004485 Application 11/629,982 case of obviousness-type double patenting, the pending claims must "read on" or be obvious in view of the claims of the copending application. As a general rule, obviousness-type double patenting determinations tum on a comparison between a patentee's earlier and later claims, with the earlier patent's written description considered only to the extent necessary to construe its claims. E.g., In re Avery, 518 F.2d 1228, 1232 [186 USPQ 161] (CCPA 1975). This is so because the non-claim portion of the earlier patent ordinarily does not qualify as prior art against the patentee and because obviousness-type double patenting is concerned with the improper extension of exclusive rights-rights conferred and defined by the claims. The focus of the obviousness-type double patenting doctrine thus rests on preventing a patentee from claiming an obvious variant of what it has previously claimed, not what it has previously disclosed. See generally Gen. Foods, 972 F.2d at 1280-82. Eli Lilly and Co. v. Teva Parenteral Medicines Inc., 689 F.3d 1368, 1378- 1379 (Fed. Cir. 2012). There is a limited exception to this customary framework. In In re Eyck, 48 F.2d 665 (CCPA 1931), our predecessor court considered obviousness-type double patenting rejections against claims to an insulated coil made up of a conductive winding material coated with an "infusible, flexible, phenol-fatty oil composition." 48 F.2d at 665. The patent applicant, Byck, had earlier obtained a patent claiming the same phenol-oil composition, and the prior art disclosed similar coils coated with other insulating compositions. Id. at 665-66. Moreover, Byck's earlier patent had discussed using his phenol-oil composition to produce adherent insulating films on metal substrates. Id. at 666. The court concluded that, in view of the prior art and Byck's earlier patent, the pending claims were drawn not to a second, distinct invention "but only ... an obvious use of the composition there patented." Id. The court explained: It would shock one's sense of justice if an inventor could receive a patent upon a composition of matter, setting out at length in the 15 Appeal2013-004485 Application 11/629,982 specification the useful purposes of such composition, manufacture and sell it to the public, and then prevent the public from making any beneficial use of such product by securing patents upon each of the uses to which it may be adapted. Id. Thus, even though Byck's earlier patent was not prior art, the court held that its disclosure of an intended use for the previously claimed phenol-oil composition could be used in the obviousness-type double patenting analysis to reject a later claim directed to that use of the same compound. Id. at 667. Eli Lilly and Co. v. Teva Parenteral Medicines Inc., 689 F.3d 1368, 1379 (Fed. Cir. 2012). Alternatively, There are [additional] "certain instances" where the specification of an earlier patent may be used in the obviousness-type double patenting analysis .... Specifically, the specification's disclosure may be used to determine whether a claim "merely define[s] an obvious variation of what is earlier disclosed and claimed," "to learn the meaning of [claim] terms," and to "interpret[] the coverage of [a] claim." Sun Pharm. Indus., Ltd v. Eli Lilly and Co., 611F.3d1381, 1387 (Fed. Cir. 2010). Thus, the Board may look to the disclosure of the '990 application for either a definition of the term "crop" as set forth in claim 1 ('990), or as to the disclosure of uses of the methods of dressing seed, therein. We further note that there is no evidence of a restriction requirement in the '990 application or in the pending application. Thus, we, under these limited circumstances, look to the disclosure of the '990 application to the uses of the penflufen compound and method of use of dressing seed disclosed therein. The '990 application defines "crops" to include rice and discloses method of treating crops and seeds, including rice seed. Page 7, 11. 12-20. 16 Appeal2013-004485 Application 11/629,982 The '990 application claims methods of treating crop seed with penflufen, and limited use of its disclosure defines that "crops" and "seeds" used in the disclosed method include rice seed. As in Ely Lilly, we agree that it would shock one's sense of justice if an inventor could receive a patent setting out at length in the specification of the '990 application methods of treating seed with penflufen and then prevent the public from making any beneficial use of such product or disclosed process by securing patents upon each of the specific seed uses to which it may be adapted. We further find that one of the natural results flowing from the dressing of seed with penflufen within the scope of claim 7 of the pending application and claim 1 of the '990 application, may be the inherent, recognized or unrecognized, result of treatment of Rhizoctonia solani infection. Furthermore, even if it was unappreciated that rice seed could be treated in view of the soy or potato seed dressed in pending claim 1 of the '990 application a nev,rly-discovered property of the prior art process cannot support a patent on that same art, is not avoided if the patentee explicitly claims that property. In other words, the mere discovery and claiming a new benefit, treatment of Rhizoctonia solani infection, of an old process (dressing a seed with the compound, penflufen, including for promotion of early emergence of certain crops) cannot render the process of dressing a seed with penflufen again patentable. Woodruff, 919 F .2d at 1578. "The general principle that a newly-discovered property of the prior art cannot support a patent on that same art is not avoided if the patentee explicitly claims that property." Abbott Labs. v. Baxter Pharm. Products, Inc., 471 F.3d 1363, 1368 (Fed. Cir. 2006). 17 Appeal2013-004485 Application 11/629,982 The obviousness-type double patenting rejection over the '990 application is affirmed for the reasons herein and of record. CONCLUSION OF LAW The cited references support the Examiner's obviousness rejection, and obviousness-type double patenting rejection over the '990 application, which are affirmed. The obviousness-type double patenting rejection over the '773 patent is reversed. AFFIRMED 18 Copy with citationCopy as parenthetical citation